Average dosage: 50-100 mg daily
Purpose: Unlocking the HPTA system after a cure
Dosage duration: up to 4 weeks
Features: strong gonadotropin stimulator, mild anti-estrogen, low toxicity
Clomifen Citrat is a widely used drug which is used to induce ovulation in women who want to have children and to treat certain disorders of the ovarian function even after stopping the birth control pill.
Clomiphene Citrate is usually prescribed to women to help ovulate.
Clomiphene citrate causes the gonadotropin-producing cells to believe that there is a lack of sex hormones.
To do this, Clomiphene binds to the steroid receptor without triggering it and thus blocks it for the corresponding steroid (testosterone or estrogen).
Clomiphene citrate activates the natural biofeedback mechanism in the brain. This activates the release of the body's own follicle stimulating hormones (FSH) such as glycoprotein.
Clomiphene citrate therefore increases the follicle-stimulating hormone and luteinizing hormone (LH), which in women leads to follicle maturation and triggering of ovulation.
In men, the luteinizing hormone stimulates the testicular cells and regulates androgen biosynthesis in the testes. This effect is particularly beneficial for the bodybuilder at the end of a steroid regimen, when the endogenous testosterone production is below average.
Would be without further intake of synthetic TestosteronenIf testosterone levels drop well below normal, the bodybuilder would lose mass and strength very quickly.
The release of the luteinizing hormone from the anterior and middle parts of the anterior pituitary lobe is controlled by the LH releasing hormone or factor from the hypothalamus.
Clomiphene gradually increases the testosterone level over the period of ingestion. Clomiphene also appears to be effective as an anti-estrogen. Most bodybuilders suffer from increased estrogen levels at the end of a regimen due to the “aromatization” of steroids.
A high level of estrogen combined with a low level of testosterone increases the risk of developing gynecomastia. This can be counteracted by taking clomiphene.